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Synthesis of cis- and trans-2-phenoxycyclopropylamines and related compounds


, : Synthesis of cis- and trans-2-phenoxycyclopropylamines and related compounds. Journal of Medicinal Chemistry 8(4): 432-439

In continuing the study of mono-amine oxidase MAO inhibitors in these laboratories, the 2-phenoxycyclo-propylamines were synthesized and found to be potent compounds. From the various intermediates, derivatives were prepared to explore their biological potentials. Also, several substituted aryloxycyclopropylamines were synthesized to determine the relationship between chemical constitution and pharmacological activity.

US$19.90

PMID: 5884163

DOI: 10.1021/jm00328a005


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